Efficient monophosphorus ligands for palladium-catalyzed miyaura borylation.
Summary of "Efficient monophosphorus ligands for palladium-catalyzed miyaura borylation."
In combination with the Bedford Pd precursor, the new biaryl monophosphorus ligand 5 was efficient for palladium-catalyzed Miyaura borylation of sterically hindered aryl bromides at low catalyst loadings.
Affiliation
Chemical Development, Boehringer Ingelheim Pharmaceuticals Inc., Ridgefield, Connecticut 06877, United States.
Journal Details
This article was published in the following journal.
Name: Organic letters
ISSN: 1523-7052
Pages: 1366-9
Links
- PubMed Source: http://www.ncbi.nlm.nih.gov/pubmed/21319836
- DOI: http://dx.doi.org/10.1021/ol2000556
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