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Halocyclization of Unsaturated Guanidines Mediated by Koser's Reagent and Lithium Halides.

08:00 EDT 22nd October 2015 | BioPortfolio

Summary of "Halocyclization of Unsaturated Guanidines Mediated by Koser's Reagent and Lithium Halides."

The synthesis of halogenated cyclic guanidines through iodine(III)-mediated umpolung of halide salts is described. Cyclic guanidines of various sizes can be obtained with generally excellent regioselectivities through either a chloro- or a bromocyclization, using Koser's reagent and the corresponding lithium salt.

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This article was published in the following journal.

Name: The Journal of organic chemistry
ISSN: 1520-6904
Pages:

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