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A Late-Stage Functionalization Approach to Derivatives of the Pyrano3,2-acarbazole Natural Products.

08:00 EDT 10th April 2019 | BioPortfolio

Summary of "A Late-Stage Functionalization Approach to Derivatives of the Pyrano3,2-acarbazole Natural Products."

Site-selective late-stage functionalizations of a pyrano[3,2-a]carbazole core related to the murrayamine natural products is reported. Specifically, selective C3 and C6 bromination has been achieved as well as C8 borylation. These functionalizations set the stage for access to a variety of natural products as well as their derivatives.

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This article was published in the following journal.

Name: The Journal of organic chemistry
ISSN: 1520-6904
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